BDBM50293940 (R)-5-Chloro-1-(1-cyclopropylethyl)-3-(2,4,5-trimethylphenylamino)pyrazin-2(1H)-one::CHEMBL564639

SMILES C[C@H](C1CC1)n1cc(Cl)nc(Nc2cc(C)c(C)cc2C)c1=O

InChI Key InChIKey=KMNGIBWEGBKKGP-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50293940   

TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50293940((R)-5-Chloro-1-(1-cyclopropylethyl)-3-(2,4,5-trime...)
Affinity DataIC50: 4.80nMAssay Description:Displacement of [125I]ovine-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed