BDBM50301787 (R)-3-methyl-6-(2-methylpiperazin-1-yl)-2-(2-(trifluoromethyl)phenethyl)pyrimidin-4(3H)-one::CHEMBL565351

SMILES C[C@@H]1CNCCN1c1cc(=O)n(C)c(CCc2ccccc2C(F)(F)F)n1

InChI Key InChIKey=OPHCHIXWIXYSNL-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50301787   

Target5-hydroxytryptamine receptor 2C(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50301787((R)-3-methyl-6-(2-methylpiperazin-1-yl)-2-(2-(trif...)
Affinity DataEC50:  64nMAssay Description:Agonist activity at human recombinant 5HT2C receptor expressed in CHO K1 cells assessed as calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed