BDBM50302995 6-(furan-2-yl)-N-(thiophen-2-ylmethyl)quinazolin-4-amine::CHEMBL566062

SMILES C(Nc1ncnc2ccc(cc12)-c1ccco1)c1cccs1

InChI Key InChIKey=DQBNMNSFJFXDRV-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50302995   

TargetDual specificity protein kinase CLK4(Human)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50302995(6-(furan-2-yl)-N-(thiophen-2-ylmethyl)quinazolin-4...)
Affinity DataIC50: 250nMAssay Description:Inhibition of Clk4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50302995(6-(furan-2-yl)-N-(thiophen-2-ylmethyl)quinazolin-4...)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of Clk4 kinase using ATP as substrate by 33P radiolabeled kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50302995(6-(furan-2-yl)-N-(thiophen-2-ylmethyl)quinazolin-4...)
Affinity DataIC50: 3.48E+3nMAssay Description:Inhibition of Dyrk1A kinase using ATP as substrate by 33P radiolabeled kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed