BDBM50306566 2-(biphenyl-4-yloxy)-N-(2-hydroxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acetamide::CHEMBL602667

SMILES CC1(C)OB(OC1(C)C)c1ccc(O)c(NC(=O)COc2ccc(cc2)-c2ccccc2)c1

InChI Key InChIKey=RGBWPLFZSXJBAE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50306566   

TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306566(2-(biphenyl-4-yloxy)-N-(2-hydroxy-5-(4,4,5,5-tetra...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed