BDBM50316299 2-Benzyl-N-(3-fluorophenyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole-8-sulfonamide::CHEMBL1099285

SMILES Fc1cccc(NS(=O)(=O)c2ccc3[nH]c4CCN(Cc5ccccc5)Cc4c3c2)c1

InChI Key InChIKey=KLXAHKWEYNGGPP-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50316299   

Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50316299(2-Benzyl-N-(3-fluorophenyl)-2,3,4,5-tetrahydro-1H-...)
Affinity DataIC50: 3.90E+3nMAssay Description:Antagonist activity at human recombinant 5HT6 receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced cAMP production by LANCE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed