BDBM50317867 4-(2-(3-tert-Butylphenylamino)ethyl)-1H-imidazole::CHEMBL1096517

SMILES CC(C)(C)c1cccc(NCCc2cnc[nH]2)c1

InChI Key InChIKey=LRIVTYQQFCXAFC-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50317867   

TargetHistamine H3 receptor(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317867(4-(2-(3-tert-Butylphenylamino)ethyl)-1H-imidazole ...)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317867(4-(2-(3-tert-Butylphenylamino)ethyl)-1H-imidazole ...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H[N-alpha-methylhistamine form human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed