BDBM50317868 4-(2-(4-tert-Butylphenylamino)ethyl)-1H-imidazole::CHEMBL1096516

SMILES CC(C)(C)c1ccc(NCCc2cnc[nH]2)cc1

InChI Key InChIKey=CAUIWLDBMLQRJD-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50317868   

TargetHistamine H3 receptor(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317868(4-(2-(4-tert-Butylphenylamino)ethyl)-1H-imidazole ...)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317868(4-(2-(4-tert-Butylphenylamino)ethyl)-1H-imidazole ...)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H[N-alpha-methylhistamine form human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed