BDBM50320258 1-(1-cyclopropylethyl)-5-(6-methoxy-2,5-dimethylpyridin-3-ylamino)-3-methyl-1,2,4-triazin-6(1H)-one::CHEMBL1084204

SMILES COc1nc(C)c(Nc2nc(C)nn(C(C)C3CC3)c2=O)cc1C

InChI Key InChIKey=UGPILKNTMDGQOW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50320258   

TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50320258(1-(1-cyclopropylethyl)-5-(6-methoxy-2,5-dimethylpy...)
Affinity DataIC50: 26nMAssay Description:Displacement of [125I]Tyr-ovine CRF from rat CRF1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed