BDBM50321576 1-(4-(3-aminoazetidine-1-carbonyl)-5-(2-fluoro-4-iodophenylamino)-1-methyl-1H-pyrrol-2-yl)ethanone::CHEMBL1172521

SMILES CC(=O)c1cc(C(=O)N2CC(N)C2)c(Nc2ccc(I)cc2F)n1C

InChI Key InChIKey=XAFMIDMQPXYJKC-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50321576   

TargetDual specificity mitogen-activated protein kinase kinase 1(Human)
Takeda California

Curated by ChEMBL

LigandBDBM50321576(1-(4-(3-aminoazetidine-1-carbonyl)-5-(2-fluoro-4-i...)Copy SMILESCopy InChI

Affinity DataIC50: 7nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
12/31/2012
Entry Details Article
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