BDBM50325811 CHEMBL1224725::N,N-dimethyl-4-(2'-(trifluoromethoxy)biphenyl-3-yl)thiazole-2-carboxamide

SMILES CN(C)C(=O)c1nc(cs1)-c1cccc(c1)-c1ccccc1OC(F)(F)F

InChI Key InChIKey=UUUHMVAHMUDADX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50325811   

TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325811(N,N-dimethyl-4-(2'-(trifluoromethoxy)biphenyl-3-yl...)
Affinity DataIC50: 1.37E+3nMAssay Description:Blockade of human Nav1.7 by voltage ion probe reader based FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed