BDBM50334726 CHEMBL1642877::N-(3-(Naphthalen-1-ylsulfonyl)-1H-indazol-7-yl)piperidine-3-carboxamide HCl

SMILES O=C(Nc1cccc2c(n[nH]c12)S(=O)(=O)c1cccc2ccccc12)C1CCCNC1

InChI Key InChIKey=YOAQEPCUBHMMFC-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50334726   

Target5-hydroxytryptamine receptor 6(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50334726(N-(3-(Naphthalen-1-ylsulfonyl)-1H-indazol-7-yl)pip...)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]-LSD from cloned human 5-HT6 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50334726(N-(3-(Naphthalen-1-ylsulfonyl)-1H-indazol-7-yl)pip...)
Affinity DataIC50: 48nMAssay Description:Antagonist activity at cloned human 5-HT6 receptor expressed in human HeLa cells assessed as inhibition of 5HT-induced cyclic AMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed