BDBM50342703 CHEMBL1771104::rac-4-(3-(2-(3-(1-(5-chloropyrimidin-2-yl)piperidin-4-yl)propyl)cyclopropyl)propoxy)-N-cyclopropyl-2-fluorobenzamide

SMILES Fc1cc(OCCCC2CC2CCCC2CCN(CC2)c2ncc(Cl)cn2)ccc1C(=O)NC1CC1

InChI Key InChIKey=UKIRDFAQOIZTRR-UHFFFAOYSA-N

Data  1 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50342703   

LigandPNGBDBM50342703(rac-4-(3-(2-(3-(1-(5-chloropyrimidin-2-yl)piperidi...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM50342703(rac-4-(3-(2-(3-(1-(5-chloropyrimidin-2-yl)piperidi...)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM50342703(rac-4-(3-(2-(3-(1-(5-chloropyrimidin-2-yl)piperidi...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed