BDBM50357608 CHEMBL1915642

SMILES CN(C)CCOc1ccc(Nc2nc3c(cccc3c3cnccc23)-c2nnc[nH]2)c(F)c1

InChI Key InChIKey=OZZCHQRAYPMEEI-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50357608   

TargetSerine/threonine-protein kinase pim-1(Human)
Zarqa University

Curated by ChEMBL
LigandPNGBDBM50357608(CHEMBL1915642)
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant PIM1 in presence of ATP by ELISA based spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Zarqa University

Curated by ChEMBL
LigandPNGBDBM50357608(CHEMBL1915642)
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant Pim1 using RSRHSSYPAGT as substrate by radiometric assay in the presence of 30 uM [ATP]More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Cylene Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357608(CHEMBL1915642)
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant Pim2 using RSRHSSYPAGT as substrate by radiometric assay in the presence of 5 uM [ATP]More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed