BDBM50364308 CHEMBL1949760

SMILES Fc1ccccc1S(=O)(=O)c1ccc2[C@@H]3CCNC[C@@H]3Oc2c1

InChI Key InChIKey=CONQSDBWMDPMKW-UHFFFAOYSA-N

Data  2 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50364308   

Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364308(CHEMBL1949760)
Affinity DataIC50: 179nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364308(CHEMBL1949760)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Rat)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364308(CHEMBL1949760)
Affinity DataKi:  145nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed