BDBM50365874 CHEMBL1957863

SMILES Cc1c(Cn2c3ccccc3n3c2nc(cc3=O)N2CCOCC2)cccc1C(F)(F)F

InChI Key InChIKey=FAIJIDJLCPUEEX-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50365874   

LigandPNGBDBM50365874(CHEMBL1957863)
Affinity DataIC50: 32nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50365874(CHEMBL1957863)
Affinity DataIC50: 80nMAssay Description:Inhibition of PI3Kdelta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50365874(CHEMBL1957863)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of PI3Kgamma by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50365874(CHEMBL1957863)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of PI3Kalpha by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed