BDBM50365880 CHEMBL1957868

SMILES CC1CN(CCO1)c1cc(=O)n2ccn(Cc3cccc(c3C)C(F)(F)F)c2n1

InChI Key InChIKey=VYOJFSXRCPAYQT-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50365880   

LigandPNGBDBM50365880(CHEMBL1957868)
Affinity DataIC50: 6nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50365880(CHEMBL1957868)
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3Kdelta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50365880(CHEMBL1957868)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of PI3Kgamma by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50365880(CHEMBL1957868)
Affinity DataIC50: 790nMAssay Description:Inhibition of PI3Kalpha by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed