BDBM50379239 CHEMBL2011477

SMILES O=C(CCCCCc1ccc(cc1)-c1ccccc1)OC[C@H]1CO1

InChI Key InChIKey=ZFBCBALKAKGXMN-UHFFFAOYSA-N

Data  12 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 12 hits for monomerid = 50379239   

TargetMonoglyceride lipase(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50379239(CHEMBL2011477)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant his-tagged MAGL expressed in Escherichia coli assessed as hydrolysis of 4-nitrophenyl acetate after 20 mins by microp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50379239(CHEMBL2011477)
Affinity DataIC50: 3.89E+3nMAssay Description:Inhibition of rat brain cytosolic MAGL assessed as [3H]-2-arachidonoyl glycerol hydrolysis after 10 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50379239(CHEMBL2011477)
Affinity DataIC50: 5.13E+3nMAssay Description:Inhibition of rat brain cytosolic MAGL assessed as [3H]-2-arachidonoyl glycerol hydrolysis after 10 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50379239(CHEMBL2011477)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant his-tagged MAGL expressed in Escherichia coli assessed as hydrolysis of 4-nitrophenyl acetate after 20 mins by microp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50379239(CHEMBL2011477)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human recombinant his-tagged MAGL expressed in Escherichia coli assessed as hydrolysis of 4-nitrophenyl acetate after 20 mins by microp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50379239(CHEMBL2011477)
Affinity DataIC50: 4.07E+3nMAssay Description:Inhibition of human recombinant his-tagged MAGL expressed in Escherichia coli assessed as hydrolysis of 4-nitrophenyl acetate after 20 mins by microp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50379239(CHEMBL2011477)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of rat brain cytosolic MAGL assessed as [3H]-2-arachidonoyl glycerol hydrolysis after 10 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50379239(CHEMBL2011477)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of rat brain membrane FAAH assessed as [3H]-anandamide hydrolysis after 10 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50379239(CHEMBL2011477)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of rat brain membrane FAAH assessed as [3H]-anandamide hydrolysis after 10 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50379239(CHEMBL2011477)
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of rat brain membrane FAAH assessed as [3H]-anandamide hydrolysis after 10 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50379239(CHEMBL2011477)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of rat brain cytosolic MAGL assessed as [3H]-2-arachidonoyl glycerol hydrolysis after 10 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50379239(CHEMBL2011477)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of rat brain membrane FAAH assessed as [3H]-anandamide hydrolysis after 10 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed