BDBM50381260 CHEMBL2018680

SMILES OC1CCN(CC1)c1nc2ccccc2nc1S(=O)(=O)c1ccc(Br)cc1

InChI Key InChIKey=RGQAORGLDQFYED-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50381260   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang University

Curated by ChEMBL

LigandBDBM50381260(CHEMBL2018680)Copy SMILESCopy InChI

Affinity DataIC50: 25nMAssay Description:Inhibition of PI3Kalpha using diC8-PI(4,5)P2 as substrate after 3 hrs by competitive fluorescence polarization assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
2/7/2013
Entry Details Article
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