BDBM50381768 CHEMBL2022867

SMILES c1nn(cc1-c1ccnc2ccccc12)-c1ccccc1

InChI Key InChIKey=GLJRDKAYQYOCDN-UHFFFAOYSA-N

Data  2 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50381768   

TargetMetabotropic glutamate receptor 4(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50381768(CHEMBL2022867)
Affinity DataEC50:  220nMAssay Description:Positive allosteric modulation of human mGlu4 receptor expressed in BHK cells assessed as potentiation of glutamate-induced calcium mobilization by F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50381768(CHEMBL2022867)
Affinity DataEC50:  920nMAssay Description:Agonist activity at MT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50381768(CHEMBL2022867)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of 5HT2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50381768(CHEMBL2022867)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human ERG by electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed