BDBM50395852 CHEMBL2165527

SMILES COc1ccc2n(c3CCC(Cc3c2c1)N(C)C)S(=O)(=O)c1ccccc1

InChI Key InChIKey=WJGHDFLJHZUCKM-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50395852   

Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandPNGBDBM50395852(CHEMBL2165527)
Affinity DataIC50: 457nMAssay Description:Antagonist activity at human recombinant 5-HT6 receptor expressed in CHO cells assessed as inhibition of 5-HT-stimulated cAMP accumulation after 4 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandPNGBDBM50395852(CHEMBL2165527)
Affinity DataKi:  5.44nMAssay Description:Displacement of [3H]LSD from human cloned 5-HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed