BDBM50405697 CHEMBL4164140

SMILES COc1ccc(cc1)-c1cc2cc(cc(C)c2oc1=O)C1Nc2ccccc2C(=O)N1C

InChI Key InChIKey=RWDKPYFVKVENAZ-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50405697   

TargetHydroxycarboxylic acid receptor 2(Human)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50405697(CHEMBL4164140)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR109a expressed in HEK293 cells harboring glosensor-22F cAMP plasmid DNA assessed as inhibition of forskolin-stimulated c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50405697(CHEMBL4164140)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR109a expressed in HEK293 cells harboring glosensor-22F cAMP plasmid DNA assessed as inhibition of forskolin-stimulated c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50405697(CHEMBL4164140)
Affinity DataEC50:  1.69E+3nMAssay Description:Agonist activity at human GPR109a expressed in HTLA cells assessed as increase in beta-arrestin2 recruitment after overnight incubation by Tango assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50405697(CHEMBL4164140)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GPR109a expressed in HTLA cells assessed as increase in beta-arrestin2 recruitment after overnight incubation by Tango assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed