BDBM50408252 CHEMBL2115488

SMILES C[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](COCc1ccccc1)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)OCc1ccccc1)C(N)=O

InChI Key InChIKey=KXDGVOMWEJNZDH-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50408252   

LigandPNGBDBM50408252(CHEMBL2115488)
Affinity DataIC50: 35nMAssay Description:Inhibitory concentration against rat brain farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
LigandPNGBDBM50408252(CHEMBL2115488)
Affinity DataIC50: 35nMAssay Description:Inhibition of rat brain farnesyltransferase in 30 mM potassium phosphate bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
LigandPNGBDBM50408252(CHEMBL2115488)
Affinity DataIC50: 102nMAssay Description:Inhibition of rat brain farnesyltransferase in 5 mM potassium phosphate and 50 mM HEPES bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
LigandPNGBDBM50408252(CHEMBL2115488)
Affinity DataIC50: 510nMAssay Description:Inhibition of rat brain farnesyltransferase in 50 mM HEPES bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed