BDBM50418186 CHEMBL1761690

SMILES CCN(Cc1c(noc1-c1ccc(cc1)C(F)(F)F)C(=O)N[C@@H]1CCC[C@H](O)C1)C(C)C

InChI Key InChIKey=DISXQTWISHCFDW-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50418186   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Msd

Curated by ChEMBL

LigandBDBM50418186(CHEMBL1761690)Copy SMILESCopy InChI

Affinity DataIC50: 25.1nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO-K1 cells assessed as inhibition of capsaicin-induced intracellular Ca2+ influx by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
5/22/2013
Entry Details Article
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