BDBM50422914 CHEMBL215932

SMILES Clc1ccc(cc1)-c1cc2ncn(-c3ccc4nc(NC5CC5)[nH]c4c3)c(=O)c2s1

InChI Key InChIKey=IZFIBMWWSGZPCL-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50422914   

TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422914(CHEMBL215932)
Affinity DataIC50: 16nMAssay Description:Antagonist activity against MCH1R expressed in CHO cells assessed as inhibition of MCH-induced EC80 thrombin response by luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed