BDBM50443637 CHEMBL3092864

SMILES NCCOCCOCCOc1ccc(NC2=NC(=Cc3ccccc3)C(=O)N2)cc1

InChI Key InChIKey=CQNULDWOIXHYFM-UHFFFAOYSA-N

Data  11 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 50443637   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50443637(CHEMBL3092864)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of human recombinant DYRK1A expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50443637(CHEMBL3092864)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant DYRK3 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50443637(CHEMBL3092864)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK9/cyclin T using YSPTSPSYSPTSPSYSPTSPSKKKK as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50443637(CHEMBL3092864)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Mouse)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50443637(CHEMBL3092864)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse recombinant CLK2 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50443637(CHEMBL3092864)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Mouse)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50443637(CHEMBL3092864)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse recombinant CLK4 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50443637(CHEMBL3092864)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant DYRK2 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50443637(CHEMBL3092864)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK2/cyclin A using [gamma-33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK3(Mouse)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50443637(CHEMBL3092864)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse recombinant CLK3 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
University of Rennes 1

Curated by ChEMBL
LigandPNGBDBM50443637(CHEMBL3092864)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant DYRK1B expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed