BDBM50444265 CHEMBL3093633

SMILES O[C@H]1CC[C@@H](CC1)Nc1nc(NCc2ccc(F)cc2)ncc1C(=O)Nc1ccc(cc1)S(=O)(=O)N1CCOCC1

InChI Key InChIKey=KNJWVKYCJCNLTC-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50444265   

TargetTyrosine-protein kinase Mer(Human)
Eshelman School of Pharmacy�Department of Pharmacology�Lineberger Compreh

Curated by ChEMBL
LigandPNGBDBM50444265(CHEMBL3093633)
Affinity DataIC50: 120nMAssay Description:Inhibition of Mer kinase (unknown origin) using 5-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by microfluidic capillary electrophoresis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Eshelman School of Pharmacy�Department of Pharmacology�Lineberger Compreh

Curated by ChEMBL
LigandPNGBDBM50444265(CHEMBL3093633)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Axl kinase (unknown origin) using 5-FAM-KKKKEEIYFFF-CONH2 as substrate after 180 mins by microfluidic capillary electrophoresis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor TYRO3(Human)
Eshelman School of Pharmacy�Department of Pharmacology�Lineberger Compreh

Curated by ChEMBL
LigandPNGBDBM50444265(CHEMBL3093633)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Tyro-3 kinase (unknown origin) using 5-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by microfluidic capillary electrophoresis as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed