BDBM50458528 CHEMBL4208934

SMILES CCc1cc(nc(n1)N1CCN(C)CC1)-c1ccoc1

InChI Key InChIKey=GOZPYYFAYISDDO-UHFFFAOYSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50458528   

Target5-hydroxytryptamine receptor 7(Human)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50458528(CHEMBL4208934)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]5-CT from human 5-HT7b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50458528(CHEMBL4208934)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A receptor expressed in HEK293 cells incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50458528(CHEMBL4208934)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50458528(CHEMBL4208934)
Affinity DataKi:  466nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cells incubated for 1 hRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50458528(CHEMBL4208934)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A expressed in HEK293 cell membranes incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed