BDBM50465617 CHEMBL4280979

SMILES OC(=O)c1ccc(CN2CCc3c([nH]c4ccccc34)C2c2ccccc2)cc1

InChI Key InChIKey=WCCPZEOFGDGTBI-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50465617   

TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Salerno

Curated by ChEMBL

LigandBDBM50465617(CHEMBL4280979)Copy SMILESCopy InChI

Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/18/2020
Entry Details Article
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