BDBM50474246 CHEMBL319658

SMILES NC[C@H]1O[C@@H](C=C1)c1c[nH]cn1

InChI Key InChIKey=DCDBUDNURLZBED-UHFFFAOYSA-N

Data  2 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50474246   

TargetHistamine H3 receptor(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474246(CHEMBL319658)
Affinity DataKi:  2.51E+3nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474246(CHEMBL319658)
Affinity DataEC50:  2.82E+3nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474246(CHEMBL319658)
Affinity DataEC50:  8.51E+4nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474246(CHEMBL319658)
Affinity DataKi: <1.00E+5nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed