BDBM50500657 CHEMBL3752106

SMILES COc1ccc(NC(=O)C2CCN(CC2)C(=O)C(C)c2ccc(CC(C)C)cc2)c(c1)[N+]([O-])=O

InChI Key InChIKey=KKEWVQGGOXZNCE-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50500657   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Henan University

Curated by ChEMBL

LigandBDBM50500657(CHEMBL3752106)Copy SMILESCopy InChI

Affinity DataIC50: 325nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
9/4/2020
Entry Details Article
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