BDBM50511114 CHEMBL4438585

SMILES CC[C@H](N1Cc2cc3O[C@@H](C(=O)N(C)c3cc2C[C@H]1C(=O)N[C@@H](Cc1ccc(cc1)-c1ccc(cc1)C#N)C(O)=O)c1ccc(OCc2ccc(Cl)c(Cl)c2)cc1)c1ccccc1

InChI Key InChIKey=ZXJQFMYVTDGFTB-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50511114   

TargetGlucagon-like peptide 1 receptor(Human)
Terns Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50511114(CHEMBL4438585)
Affinity DataEC50:  59nMAssay Description:Displacement of [125I]GLP-1 from human GLP-1R (7 to 36 residues) expressed in HEK293 or CHO cell membranes after 120 mins by radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed