BDBM50520815 CHEMBL4574711

SMILES CCCCC[C@@H](O)c1nc(-c2ccccc2)n(c1\C=C\[C@@H](O)[C@@H](O)CCCC(=O)OC)-c1ccccc1

InChI Key InChIKey=VGXMROVCMLMHKD-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50520815   

TargetN-formyl peptide receptor 2(Human)
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50520815(CHEMBL4574711)
Affinity DataIC50: 0.5nMAssay Description:Agonist activity at ALX/FPR2 in human THP1 cells harboring NF-kB-Luc assessed as inhibition of LPS-induced NFkB signalling activation by measuring re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetN-formyl peptide receptor 2(Human)
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50520815(CHEMBL4574711)
Affinity DataIC50: 1.40nMAssay Description:Agonist activity at ALX/FPR2 in human THP1 cells harboring NF-kB-Luc assessed as inhibition of LPS-induced NFkB signalling activation by measuring re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetN-formyl peptide receptor 2(Human)
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50520815(CHEMBL4574711)
Affinity DataIC50: 7.10nMAssay Description:Agonist activity at ALX/FPR2 in human THP1 cells harboring NF-kB-Luc assessed as inhibition of LPS-induced NFkB signalling activation by measuring re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetN-formyl peptide receptor 2(Human)
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50520815(CHEMBL4574711)
Affinity DataIC50: 10nMAssay Description:Agonist activity at ALX/FPR2 in human THP1 cells harboring NF-kB-Luc assessed as inhibition of LPS-induced NFkB signalling activation by measuring re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetN-formyl peptide receptor 2(Human)
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50520815(CHEMBL4574711)
Affinity DataIC50: 19nMAssay Description:Agonist activity at ALX/FPR2 in human THP1 cells harboring NF-kB-Luc assessed as inhibition of LPS-induced NFkB signalling activation by measuring re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetN-formyl peptide receptor 2(Human)
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50520815(CHEMBL4574711)
Affinity DataIC50: 26nMAssay Description:Agonist activity at ALX/FPR2 in human THP1 cells harboring NF-kB-Luc assessed as inhibition of LPS-induced NFkB signalling activation pretreated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed