BDBM50521261 CHEMBL4584670

SMILES COC(=O)C1CN(C1)c1ccc(cn1)N1CC[C@@H](Oc2ccc(OCC(F)(F)F)nc2)C1=O

InChI Key InChIKey=KAAXJOJIEQSMGS-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50521261   

TargetGlucose-dependent insulinotropic receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50521261(CHEMBL4584670)
Affinity DataEC50:  12nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as intracellular cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed