BDBM50521885 CHEMBL4459061

SMILES CC1CN(C(=O)Cc2nc3nc(C)cc(C)n3n2)c2nc3ccccc3n12

InChI Key InChIKey=CHJKSRSGLBJMRH-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50521885   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50521885(CHEMBL4459061)Copy SMILESCopy InChI

Affinity DataIC50: 292nMAssay Description:Inhibition of human PDE10A using cAMP as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by HTRF detecti...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/23/2021
Entry Details Article
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