BDBM50521998 CHEMBL4450094

SMILES COc1cc(OC)cc(c1)C(=O)Nc1nc(c(CCCN2CCN(C)CC2)s1)-c1ccccc1

InChI Key InChIKey=DMRMHEZQZBDALQ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50521998   

TargetTransient receptor potential cation channel subfamily V member 4(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50521998(CHEMBL4450094)Copy SMILESCopy InChI

Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human TRPV4 expressed in HEK293 cells assessed as reduction in Ca2+ influx incubated for 30 mins by Fluo4-AM dye basedMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/23/2021
Entry Details Article
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