BDBM50522000 CHEMBL4586243

SMILES COc1cc(OC)cc(c1)C(=O)Nc1nc(c(CCCN(C)C)s1)-c1ccccc1

InChI Key InChIKey=MYPKRCJGRKTUFB-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50522000   

TargetTransient receptor potential cation channel subfamily V member 4(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50522000(CHEMBL4586243)Copy SMILESCopy InChI

Affinity DataIC50: 86nMAssay Description:Inhibition of human TRPV4 expressed in HEK293 cells assessed as reduction in Ca2+ influx incubated for 30 mins by Fluo4-AM dye basedMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/23/2021
Entry Details Article
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