BDBM50522718 CHEMBL4513964

SMILES CC(C)(C)c1ccc(cc1)-c1ccc2n(ncc2c1)C(CC1CCCCC1)c1ccc(cc1)C(=O)NCCC(O)=O

InChI Key InChIKey=AOYSALLRSAQXLS-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50522718   

TargetGlucagon receptor(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50522718(CHEMBL4513964)
Affinity DataKi:  114nMAssay Description:Antagonist activity at full length human recombinant GCGR transfected in HEK293 cells assessed as inhibition of glucagon-stimulated cAMP by by LANCE ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed