BDBM50522727 CHEMBL4441433

SMILES CC(C)CC(c1ccc(cc1)C(=O)NCCC(O)=O)n1ncc2cc(ccc12)-c1ccc(cc1)N1CCN(C)CC1

InChI Key InChIKey=CXBZJHBWNIPARM-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50522727   

TargetGlucagon receptor(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50522727(CHEMBL4441433)
Affinity DataKi:  1.25E+3nMAssay Description:Antagonist activity at full length human recombinant GCGR transfected in HEK293 cells assessed as inhibition of glucagon-stimulated cAMP by by LANCE ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed