BDBM50524377 CHEMBL4519923

SMILES CCCCc1cc(nc(N)n1)-c1ccc(OC)cc1

InChI Key InChIKey=NGUDUTAVPODMJD-UHFFFAOYSA-N

Data  2 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50524377   

TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524377(CHEMBL4519923)
Affinity DataIC50: 4.47E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524377(CHEMBL4519923)
Affinity DataEC50:  5.18E+3nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524377(CHEMBL4519923)
Affinity DataIC50: 4.45E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524377(CHEMBL4519923)
Affinity DataEC50:  5.25E+3nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed