BDBM50526164 CHEMBL4589724

SMILES Nc1ccccc1NC(=O)c1cnc(NCc2ccccc2)cn1

InChI Key InChIKey=VNDKSSOLKIUTSX-UHFFFAOYSA-N

Data  11 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 50526164   

TargetHistone deacetylase 3(Human)
Birla Institute of Technology and Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50526164(CHEMBL4589724)
Affinity DataIC50: 245nMAssay Description:Inhibition of recombinant human HDAC3 using fluorescent as substrate measured for 15 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Birla Institute of Technology and Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50526164(CHEMBL4589724)
Affinity DataIC50: 245nMAssay Description:Inhibition of human recombinant HDAC3 incubated for 15 mins by fluorescence based microplate analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Birla Institute of Technology and Science-Pilani Hyderabad

Curated by ChEMBL
LigandPNGBDBM50526164(CHEMBL4589724)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human recombinant HDAC1 incubated for 15 mins by fluorescence based microplate analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Birla Institute of Technology and Science-Pilani Hyderabad

Curated by ChEMBL
LigandPNGBDBM50526164(CHEMBL4589724)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of recombinant human HDAC1 using fluorescent as substrate measured for 15 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetHistone deacetylase 8(Human)
Birla Institute of Technology and Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50526164(CHEMBL4589724)
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of recombinant human HDAC8 using fluorescent as substrate measured for 10 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetHistone deacetylase 2(Human)
Birla Institute of Technology and Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50526164(CHEMBL4589724)
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of recombinant human HDAC2 using fluorescent as substrate measured for 30 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetHistone deacetylase 2(Human)
Birla Institute of Technology and Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50526164(CHEMBL4589724)
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of human recombinant HDAC2 incubated for 30 mins by fluorescence based microplate analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Birla Institute of Technology and Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50526164(CHEMBL4589724)
Affinity DataIC50: 3.72E+3nMAssay Description:Inhibition of recombinant human HDAC6 using fluorescent as substrate measured for 10 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetHistone deacetylase 8(Human)
Birla Institute of Technology and Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50526164(CHEMBL4589724)
Affinity DataIC50: 1.56E+4nMAssay Description:Inhibition of human recombinant HDAC8 incubated for 10 mins by fluorescence based microplate analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Birla Institute of Technology and Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50526164(CHEMBL4589724)
Affinity DataIC50: 3.72E+4nMAssay Description:Inhibition of human recombinant HDAC6 incubated for 15 mins by fluorescence based microplate analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetNuclear receptor corepressor 1(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50526164(CHEMBL4589724)
Affinity DataIC50: 6.56E+4nMAssay Description:Inhibition of human recombinant HDAC3/GST-tagged NCOR1 DAD (397 to 503 residues) expressed in baculovirus expression system using Fluor de Lys as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed