BDBM50532409 CHEMBL4445077

SMILES CC(C)C[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)C\C=C/C[C@H](N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O

InChI Key InChIKey=YSFKNPRFMZPTER-UHFFFAOYSA-N

Data  4 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50532409   

TargetNeuropeptide Y receptor type 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50532409(CHEMBL4445077)
Affinity DataEC50:  30nMAssay Description:Agonist activity at GFP-tagged neuropeptide Y4R (unknown origin) expressed in HEK293T cells assessed as beta-arrestin2 recruitment measured after 60 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50532409(CHEMBL4445077)
Affinity DataEC50:  30nMAssay Description:Agonist activity at GFP-tagged neuropeptide Y4R (unknown origin) expressed in HEK293T cells assessed as beta-arrestin2 recruitment measured after 60 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50532409(CHEMBL4445077)
Affinity DataIC50: 132nMAssay Description:Displacement of [Lys2(sCy5),Arg4]-BVD-15 from C-terminal GFP-tagged neuropeptide Y4R (unknown origin) expressed in human 293TR cells measured after 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50532409(CHEMBL4445077)
Affinity DataIC50: 132nMAssay Description:Displacement of [Lys2(sCy5),Arg4]-BVD-15 from C-terminal GFP-tagged neuropeptide Y4R (unknown origin) expressed in human 293TR cells measured after 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50532409(CHEMBL4445077)
Affinity DataIC50: 490nMAssay Description:Agonist activity at GFP-tagged neuropeptide Y1R (unknown origin) expressed in HEK293T cells assessed as beta-arrestin2 recruitment measured after 60 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50532409(CHEMBL4445077)
Affinity DataIC50: 490nMAssay Description:Agonist activity at GFP-tagged neuropeptide Y1R (unknown origin) expressed in HEK293T cells assessed as beta-arrestin2 recruitment measured after 60 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed