BDBM50537001 CHEMBL4520937

SMILES CCn1c2ccc(cc2c2cccc(C)c12)-c1nc2c(C)c(ccc2n1CCOC)C(O)=O

InChI Key InChIKey=RCRVYFOWDPTKSK-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50537001   

TargetProstaglandin E2 receptor EP4 subtype(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50537001(CHEMBL4520937)
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity at human EP4R assessed as inhibition of agonist-induced cAMP production by fluorescent cAMP tracer cAMP-d2 based FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed