BDBM50558283 CHEMBL4758929

SMILES CO[C@@H]1CCN(C1)c1ccc(Cc2cc(C(=O)N[C@H]3CCCC[C@@H]3O)c(=O)n(C)c2C)cc1

InChI Key InChIKey=QIKBSXNGZUTBFE-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50558283   

TargetMuscarinic acetylcholine receptor M1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50558283(CHEMBL4758929)
Affinity DataEC50:  1.69E+3nMAssay Description:Positive allosteric modulation of human muscarinic M1 receptor stably expressed in CHO cells assessed as increase in Ach-induced intracellular calciu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed