BDBM50559212 CHEMBL4797000

SMILES Fc1ccc(CNC(=O)Cc2nnc(o2)-c2ccc3OCOc3c2)cc1

InChI Key InChIKey=HFYXIEMXPIVPKY-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50559212   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang University

Curated by ChEMBL

LigandBDBM50559212(CHEMBL4797000)Copy SMILESCopy InChI

Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2 as substrate measured after 1 hr by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
3/27/2022
Entry Details Article
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