BDBM50564969 CHEMBL4799113

SMILES COCC\C(Nc1ccc(Oc2ccnc3cc(OCCCN4CCOCC4)c(OC)cc23)c(F)c1)=N/S(=O)(=O)Cc1ccc(Cl)cc1

InChI Key InChIKey=QCKKTDVCCCBGDD-UHFFFAOYSA-N

Data  10 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 50564969   

TargetHepatocyte growth factor receptor(Human)
Harbin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50564969(CHEMBL4799113)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of c-MET (unknown origin) using poly (Glu, Tyr)4:1 as substrate in presence of ATP measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Harbin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50564969(CHEMBL4799113)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of c-Kit (unknown origin) using poly (Glu, Tyr)4:1 as substrate in presence of ATP measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor alpha(Human)
Harbin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50564969(CHEMBL4799113)
Affinity DataIC50: 384nMAssay Description:Inhibition of PDGFR alpha (unknown origin) using poly (Glu, Tyr)4:1 as substrate in presence of ATP measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Harbin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50564969(CHEMBL4799113)
Affinity DataIC50: 565nMAssay Description:Inhibition of PDGFR beta (unknown origin) using poly (Glu, Tyr)4:1 as substrate in presence of ATP measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Harbin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50564969(CHEMBL4799113)
Affinity DataIC50: 412nMAssay Description:Inhibition of Ron (unknown origin) using poly (Glu, Tyr)4:1 as substrate in presence of ATP measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Harbin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50564969(CHEMBL4799113)
Affinity DataIC50: 673nMAssay Description:Inhibition of VEGFR 2 (unknown origin) using poly (Glu, Tyr)4:1 as substrate in presence of ATP measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Harbin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50564969(CHEMBL4799113)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of EGFR (unknown origin) using poly (Glu, Tyr)4:1 as substrate in presence of ATP measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Harbin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50564969(CHEMBL4799113)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of FLT-3 (unknown origin) using poly (Glu, Tyr)4:1 as substrate in presence of ATP measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Harbin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50564969(CHEMBL4799113)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ALK (unknown origin) using poly (Glu, Tyr)4:1 as substrate in presence of ATP measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 3(Human)
Harbin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50564969(CHEMBL4799113)
Affinity DataIC50: 358nMAssay Description:Inhibition of FLT-4 (unknown origin) using poly (Glu, Tyr)4:1 as substrate in presence of ATP measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed