BDBM50595436 CHEMBL5177502

SMILES OC[C@H]1O[C@H]([C@H](O)[C@@H](O)[C@@H]1O)c1ccc(Cl)c(Cc2ccc(OC3CCOC3)cc2)c1

InChI Key InChIKey=OBWASQILIWPZMG-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50595436   

TargetSodium/glucose cotransporter 2(Human)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50595436(CHEMBL5177502)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cell membrane assessed as inhibition of [14C]AMG uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50595436(CHEMBL5177502)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cell membrane assessed as inhibition of [14C]AMG uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed