BDBM50596123 CHEMBL5176894

SMILES COc1ccc(\C=C2/SC(=S)NC2=O)cc1C#C[Si](C)(c1ccccc1)c1ccccc1

InChI Key InChIKey=BJFBLDLNIQFERR-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50596123   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Shinshu University

Curated by ChEMBL

LigandBDBM50596123(CHEMBL5176894)Copy SMILESCopy InChI

Affinity DataIC50: 530nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
6/22/2023
Entry Details
Copy BDB DOIPubMed
Copy reaction URL