BDBM50596124 CHEMBL5173788

SMILES COc1ccc(\C=C2/SC(=S)NC2=O)cc1C#C[Si](c1ccccc1)(c1ccccc1)c1ccccc1

InChI Key InChIKey=SKMFCQXTDNKDES-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50596124   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Shinshu University

Curated by ChEMBL

LigandBDBM50596124(CHEMBL5173788)Copy SMILESCopy InChI

Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
6/22/2023
Entry Details
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