BDBM50597584 CHEMBL5192578

SMILES Fc1ccc2c(Cc3nncn3CCCc3c[nH]cn3)c[nH]c2c1

InChI Key InChIKey=IKILUYGGNRRSKR-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50597584   

TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597584(CHEMBL5192578)
Affinity DataEC50:  1.04E+3nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597584(CHEMBL5192578)
Affinity DataKi:  717nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 2(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597584(CHEMBL5192578)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST2A receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed