BDBM50604149 CHEMBL5196648

SMILES Fc1ccc(cc1)-c1csc(n1)[C@@H]1CCCN1C(=O)Nc1cccc2cnccc12

InChI Key InChIKey=ZYAXGEGPABHQEK-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50604149   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Henan University

Curated by ChEMBL

LigandBDBM50604149(CHEMBL5196648)Copy SMILESCopy InChI

Affinity DataIC50: 24nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced Ca2+ influx incubated for 30 mins by FLIPR meth...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
6/25/2023
Entry Details
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